Parallel copper catalysis: Diastereoselective synthesis of polyfunctionalized azetidin-2-imines

Yanpeng Xing; Hongyang Zhao; Qiongyi Shang; Jing Wang; Ping Lu; Yanguang Wang

doi:10.1021/ol4010323

Parallel copper catalysis: Diastereoselective synthesis of polyfunctionalized azetidin-2-imines

Yanpeng Xing
, Hongyang Zhao
, Qiongyi Shang
, Jing Wang
, Ping Lu^*
, Yanguang Wang

^*此作品的通讯作者

Zhejiang University

科研成果: 期刊稿件 › 文章 › 同行评审

38 引用（Scopus）

摘要

An efficient and diastereoselective synthesis of highly functionalized azetidin-2-imines has been achieved through a parallel catalysis strategy, including a copper-catalyzed azide-alkyne cycloaddition, a copper-catalyzed C_sp-Csp² cross-coupling reaction, and an intermolecular [2 + 2] cycloaddition. The products could be conveniently converted into the structurally interesting dihydroazeto[1,2-a]benzo[e]azepin-2(4H)-imines.

源语言	英语
页（从-至）	2668-2671
页数	4
期刊	Organic Letters
卷	15
期	11
DOI	https://doi.org/10.1021/ol4010323
出版状态	已出版 - 7 6月 2013
已对外发布	是

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abstract = "An efficient and diastereoselective synthesis of highly functionalized azetidin-2-imines has been achieved through a parallel catalysis strategy, including a copper-catalyzed azide-alkyne cycloaddition, a copper-catalyzed Csp-Csp2 cross-coupling reaction, and an intermolecular [2 + 2] cycloaddition. The products could be conveniently converted into the structurally interesting dihydroazeto[1,2-a]benzo[e]azepin-2(4H)-imines.",

author = "Yanpeng Xing and Hongyang Zhao and Qiongyi Shang and Jing Wang and Ping Lu and Yanguang Wang",

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T1 - Parallel copper catalysis

T2 - Diastereoselective synthesis of polyfunctionalized azetidin-2-imines

AU - Xing, Yanpeng

AU - Zhao, Hongyang

AU - Shang, Qiongyi

AU - Wang, Jing

AU - Lu, Ping

AU - Wang, Yanguang

PY - 2013/6/7

Y1 - 2013/6/7

N2 - An efficient and diastereoselective synthesis of highly functionalized azetidin-2-imines has been achieved through a parallel catalysis strategy, including a copper-catalyzed azide-alkyne cycloaddition, a copper-catalyzed Csp-Csp2 cross-coupling reaction, and an intermolecular [2 + 2] cycloaddition. The products could be conveniently converted into the structurally interesting dihydroazeto[1,2-a]benzo[e]azepin-2(4H)-imines.

AB - An efficient and diastereoselective synthesis of highly functionalized azetidin-2-imines has been achieved through a parallel catalysis strategy, including a copper-catalyzed azide-alkyne cycloaddition, a copper-catalyzed Csp-Csp2 cross-coupling reaction, and an intermolecular [2 + 2] cycloaddition. The products could be conveniently converted into the structurally interesting dihydroazeto[1,2-a]benzo[e]azepin-2(4H)-imines.

UR - https://www.scopus.com/pages/publications/84879205734

U2 - 10.1021/ol4010323

DO - 10.1021/ol4010323

M3 - Article

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SN - 1523-7060

VL - 15

SP - 2668

EP - 2671

JO - Organic Letters

JF - Organic Letters

IS - 11

ER -

Parallel copper catalysis: Diastereoselective synthesis of polyfunctionalized azetidin-2-imines

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